SBR00098

Tazemetostat

≥98% (HPLC), powder

• 동의어(들): EPZ6438
• 실험식(Hill 표기법): C₃₄H₄₄N₄O₄
• CAS Number: 1403254-99-8
• Molecular Weight: 572.74
• UNSPSC 코드: 51101500

속성

• Quality Level: 100
• 분석: ≥98% (HPLC)
• 양식: powder
• 색상: white to off-white
• 동작 모드: protein synthesis | inhibits
• 저장 온도: 2-30°C
• SMILES string: CCN(C1CCOCC1)C2=CC(=CC(=C2C)C(=O)NCC3=C(C=C(NC3=O)C)C)C4=CC=C(C=C4)CN5CCOCC5
• InChI: InChI=1S/C34H44N4O4/c1-5-38(29-10-14-41-15-11-29)32-20-28(27-8-6-26(7-9-27)22-37-12-16-42-17-13-37)19-30(25(32)4)33(39)35-21-31-23(2)18-24(3)36-34(31)40/h6-9,18-20,29H,5,10-17,21-22H2,1-4H3,(H,35,39)(H,36,40)
• InChI key: NSQSAUGJQHDYNO-UHFFFAOYSA-N

설명

일반 설명

Tazemetostat is a small molecule inhibitor of the EZH2 protein, which is a histone-lysine N-methyltransferase enzyme that plays a key role in epigenetic regulation of gene expression.

생화학적/생리학적 작용

Tazemetostat inhibits the EZH2 protein. EZH2 is a histone-lysine N-methyltransferase enzyme that plays a key role in epigenetic regulation of gene expression in cells. As an epigenetic modifier, EZH2 protein controls the transcriptional repression of various genes involved in cell cycle regulation, DNA repair, and other cellular processes.

안전성 정보

• Storage Class Code: 11 - Combustible Solids
• WGK: WGK 3
• Flash Point (°F): Not applicable
• Flash Point (°C): Not applicable