A6226
AM251
>98% (HPLC), solid, cannabinoid receptor (CB1) antagonist
동의어(들):
1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide
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모든 사진(1)
About This Item
실험식(Hill 표기법):
C22H21N4OCl2I
CAS Number:
Molecular Weight:
555.24
MDL number:
UNSPSC 코드:
12352200
PubChem Substance ID:
NACRES:
NA.77
추천 제품
제품명
AM251, >98% (HPLC), solid
Quality Level
분석
>98% (HPLC)
양식
solid
색상
white
solubility
DMSO: >10 mg/mL
H2O: insoluble
주관자
Sanofi Aventis
SMILES string
Cc1c(nn(-c2ccc(Cl)cc2Cl)c1-c3ccc(I)cc3)C(=O)NN4CCCCC4
InChI
1S/C22H21Cl2IN4O/c1-14-20(22(30)27-28-11-3-2-4-12-28)26-29(19-10-7-16(23)13-18(19)24)21(14)15-5-8-17(25)9-6-15/h5-10,13H,2-4,11-12H2,1H3,(H,27,30)
InChI key
BUZAJRPLUGXRAB-UHFFFAOYSA-N
유전자 정보
mouse ... Cnr1(12801) , Cnr2(12802)
rat ... Cnr1(25248)
애플리케이션
AM251, a CB1 cannabinoid receptor antagonist, has been used in a study to determine its interaction with hippocampal neurons to enhance spatial memory in mice.
생화학적/생리학적 작용
AM251 is a CB1 cannabinoid receptor antagonist.
특징 및 장점
This compound is featured on the Cannabinoid Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.
This compound was developed by Sanofi Aventis. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.
기타 정보
Salt content may vary.
유해 및 위험 성명서
예방조치 성명서
Hazard Classifications
Aquatic Chronic 4
Storage Class Code
11 - Combustible Solids
WGK
WGK 3
Flash Point (°F)
Not applicable
Flash Point (°C)
Not applicable
개인 보호 장비
dust mask type N95 (US), Eyeshields, Gloves
이미 열람한 고객
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